Research Index

Melanotan II Research Index

PSI surfaces 50 peer-reviewed studies on Melanotan II, prioritized by evidence strength: human clinical research first, then animal studies. The full historical archive is linked below on PubMed.

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50 studies

Changes in Oral Mucosa Associated with Melanotan II Injections: A Case Report.

Bonchev A

Life (Basel)·2026·Human·PubMed →

Melanotan II nasal spray: a possible risk factor for oral mucosal malignant melanoma?

Yassin Alsabbagh A, Bhujel N, Singh RP

Int J Oral Maxillofac Surg·2025·Animal·PubMed →

Trending on TikTok: An analysis of melanotan content on social media.

Herlihy M, Bowe S, Ahmad K

J Eur Acad Dermatol Venereol·2025·Animal·PubMed →

The 'Barbie Drug'-marketing and perceptions of melanotan on social media.

Orr E, Grechin C, Kearney N et al.

J Eur Acad Dermatol Venereol·2025·Animal·PubMed →

Antidepressant-like and antistress effects of the ACTH(4-10) synthetic analogs Semax and Melanotan II on male rats in a model of chronic unpredictable stress.

Inozemtseva LS, Yatsenko KA, Glazova NY et al.

Eur J Pharmacol·2024·Animal·Anxiety & Mood·PubMed →

Barbie drug identification: Not a child's play.

Deville M, Charlier C

J Forensic Sci·2024·Animal·PubMed →

Recommended Tool Compounds for the Melanocortin Receptor (MCR) G Protein-Coupled Receptors (GPCRs).

Weirath NA, Haskell-Luevano C

ACS Pharmacol Transl Sci·2024·Animal·PubMed →

Therapeutic Strategies Against Metabolic Imbalance in a Male Mouse Model With 5-HT2CR Loss-of-Function.

Liu H, Liu Z, Wong HK et al.

Endocrinology·2024·Animal·Weight Loss, Neuroprotection·PubMed →

Multiple metabolic signals in the CeA regulate feeding: The role of AMPK.

Castro G, Mendes NF, Weissmann L et al.

Mol Cell Endocrinol·2024·Animal·PubMed →

5-Hydroxypyrroloindoline Affords Tryptathionine and 2,2'-bis-Indole Peptide Staples: Application to Melanotan-II.

Todorovic M, Blanc A, Wang Z et al.

Chemistry·2024·Animal·PubMed →

Melanocortin agonism in a social context selectively activates nucleus accumbens in an oxytocin-dependent manner.

Ford CL, McDonough AA, Horie K et al.

Neuropharmacology·2024·Animal·PubMed →

Effects of the central melanocortin system on feed intake, metabolic hormones and insulin action in the sheep.

Ehrhardt RA, Giesy SL, Hileman SM et al.

J Anim Sci·2023·Animal·PubMed →

Melanotan-II reverses memory impairment induced by a short-term HF diet.

Wekwejt P, Wojda U, Kiryk A

Biomed Pharmacother·2023·Animal·PubMed →

Obesity medication lorcaserin activates brainstem GLP-1 neurons to reduce food intake and augments GLP-1 receptor agonist induced appetite suppression.

Wagner S, Brierley DI, Leeson-Payne A et al.

Mol Metab·2023·Animal·Neuroprotection, Appetite Regulation, Weight Loss·PubMed →

Melanocortin receptor agonist melanotan-II microinjected in the nucleus accumbens decreases appetitive and consumptive responding for food.

Eliason NL, Martin L, Low MJ et al.

Neuropeptides·2022·Animal·Weight Loss·PubMed →

Vasopressin neurons in the paraventricular hypothalamus promote wakefulness via lateral hypothalamic orexin neurons.

Islam MT, Rumpf F, Tsuno Y et al.

Curr Biol·2022·Animal·Neuroprotection, Sleep·PubMed →

[The risks of tanning with the Barbie drug].

Eijmael MJPM, Janmaat CJ, Briët-Schipper EMN

Ned Tijdschr Geneeskd·2022·Animal·PubMed →

CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists.

Tomassi S, Dimmito MP, Cai M et al.

J Med Chem·2022·Animal·PubMed →

Zebrafish Bioassay for Screening Therapeutic Candidates Based on Melanotrophic Activity.

Hong TI, Hwang KS, Choi TI et al.

Int J Mol Sci·2021·Animal·PubMed →

Melanotan II User Experience: A Qualitative Study of Online Discussion Forums.

Gilhooley E, Daly S, McKenna D

Dermatology·2021·Animal·PubMed →

Depletion of Alpha-Melanocyte-Stimulating Hormone Induces Insatiable Appetite and Gains in Energy Reserves and Body Weight in Zebrafish.

Hsieh YW, Tsai YW, Lai HH et al.

Biomedicines·2021·Animal·PubMed →

Intracerebroventricular administration of α-melanocyte-stimulating hormone (α-MSH) enhances thigmotaxis and induces anxiety-like behavior in the goldfish Carassius auratus.

Watanabe K, Konno N, Nakamachi T et al.

Peptides·2021·Animal·Anxiety & Mood·PubMed →

The Mesencephalic Trigeminal Nucleus Controls Food Intake and Body Weight via Hindbrain POMC Projections.

Fortin SM, Chen J, Grill HJ et al.

Nutrients·2021·Animal·Appetite Regulation, Weight Loss, Neuroprotection·PubMed →

Melanocortin receptor activation alleviates amyloid pathology and glial reactivity in an Alzheimer's disease transgenic mouse model.

Lau JKY, Tian M, Shen Y et al.

Sci Rep·2021·Animal·Neuroprotection·PubMed →

Restoration of Cardiac Function After Myocardial Infarction by Long-Term Activation of the CNS Leptin-Melanocortin System.

Gava FN, da Silva AA, Dai X et al.

JACC Basic Transl Sci·2021·Animal·PubMed →

Melanotan Tanning Injection: A Rare Cause of Priapism.

Mallory CW, Lopategui DM, Cordon BH

Sex Med·2021·Animal·PubMed →

Pharmacological chaperone action in humanized mouse models of MC4R-linked obesity.

René P, Lanfray D, Richard D et al.

JCI Insight·2021·Animal·Glycemic Control, Weight Loss·PubMed →

Melanotan II, a melanocortin agonist, partially rescues the impaired thermogenic capacity of pituitary adenylate cyclase-activating polypeptide deficient mice.

McMillan TR, Forster MAM, Short LI et al.

Exp Physiol·2021·Animal·PubMed →

LC-HRMS characterization of the skin pigmentation and sexual enhancers melanotan II and bremelanotide sold on the black market of performance and image enhancing drugs.

Mestria S, Odoardi S, Frison G et al.

Drug Test Anal·2021·Animal·PubMed →

G(q)α/G(11)α deficiency in dorsomedial hypothalamus leads to obesity resulting from decreased energy expenditure and impaired sympathetic nerve activity.

Wilson EA, Sun H, Cui Z et al.

Am J Physiol Endocrinol Metab·2021·Animal·Weight Loss·PubMed →

A sentinel population: The public health benefits of monitoring enhanced body builders.

McVeigh J, Salinas M, Ralphs R

Int J Drug Policy·2021·Animal·PubMed →

Melanotan II: a possible cause of renal infarction: review of the literature and case report.

Peters B, Hadimeri H, Wahlberg R et al.

CEN Case Rep·2020·Human·PubMed →

Development of Ligand-Drug Conjugates Targeting Melanoma through the Overexpressed Melanocortin 1 Receptor.

Zhou Y, Mowlazadeh Haghighi S, Liu Z et al.

ACS Pharmacol Transl Sci·2020·Animal·PubMed →

CAPS2 deficiency induces proopiomelanocortin accumulation in pituitary and affects food intake behavior in mice.

Fujima S, Amemiya N, Arima T et al.

Neurosci Lett·2020·Animal·Weight Loss, Neuroprotection·PubMed →

Combining MALDI mass spectrometry imaging and droplet-base surface sampling analysis for tissue distribution, metabolite profiling, and relative quantification of cyclic peptide melanotan II.

Chen B, Vavrek M, Gundersdorf R et al.

Anal Chim Acta·2020·Animal·PubMed →

Hypothalamic POMC deficiency increases circulating adiponectin despite obesity.

Yu H, Chhabra KH, Thompson Z et al.

Mol Metab·2020·Animal·Neuroprotection, Weight Loss·PubMed →

Melanocortin regulation of histaminergic neurons via perifornical lateral hypothalamic melanocortin 4 receptors.

Michael NJ, Caron A, Lee CE et al.

Mol Metab·2020·Animal·Neuroprotection·PubMed →

Application of Dimedone Enamines as Protecting Groups for Amines and Peptides.

Chithanna S, Vyasamudri S, Yang DY

Org Lett·2020·Animal·PubMed →

Topical MTII Therapy Suppresses Melanoma Through PTEN Upregulation and Cyclooxygenase II Inhibition.

Wu JC, Tsai HE, Hsiao YH et al.

Int J Mol Sci·2020·Animal·PubMed →

Sites and sources of sympathoexcitation in obese male rats: role of brain insulin.

Shi Z, Zhao D, Cassaglia PA et al.

Am J Physiol Regul Integr Comp Physiol·2020·Animal·Weight Loss·PubMed →

Hypothalamic C2-domain protein involved in MC4R trafficking and control of energy balance.

Gavini CK, Cook TM, Rademacher DJ et al.

Metabolism·2020·Animal·Weight Loss·PubMed →

Melanotan-II reverses autistic features in a maternal immune activation mouse model of autism.

Minakova E, Lang J, Medel-Matus JS et al.

PLoS One·2019·Animal·PubMed →

Glucose-regulated protein 78 binds to and regulates the melanocortin-4 receptor.

Yoon YR, Lee TG, Choi MH et al.

Exp Mol Med·2018·Animal·Weight Loss·PubMed →

A glimpse into the underground market of melanotan.

Callaghan Iii DJ

Dermatol Online J·2018·Animal·PubMed →

Limiting feeding to the active phase reduces blood pressure without the necessity of caloric reduction or fat mass loss.

Cote I, Toklu HZ, Green SM et al.

Am J Physiol Regul Integr Comp Physiol·2018·Animal·Weight Loss·PubMed →

Melanotan II causes hypothermia in mice by activation of mast cells and stimulation of histamine 1 receptors.

Jain S, Panyutin A, Liu N et al.

Am J Physiol Endocrinol Metab·2018·Animal·PubMed →

The stimulatory G protein G(s)α is required in melanocortin 4 receptor-expressing cells for normal energy balance, thermogenesis, and glucose metabolism.

Podyma B, Sun H, Wilson EA et al.

J Biol Chem·2018·Animal·Weight Loss·PubMed →

Inherently Lean Rats Have Enhanced Activity and Skeletal Muscle Response to Central Melanocortin Receptors.

Gavini CK, Britton SL, Koch LG et al.

Obesity (Silver Spring)·2018·Animal·Muscle Recovery·PubMed →

Changes of melanocytic lesions inducedby Melanotan injections and sun bed use ina teenage patient with FAMMM syndrome.

Sivyer GW

Dermatol Pract Concept·2012·Human·PubMed →

Effect of MELANOTAN, [Nle(4), D-Phe(7)]-alpha-MSH, on melanin synthesis in humans with MC1R variant alleles.

Fitzgerald LM, Fryer JL, Dwyer T et al.

Peptides·2006·Human·PubMed →